5-Sulfoisophthalic acid | CAS:22326-31-4
5-Sulfoisophthalic acid
- 名称:5-磺酸基间苯二甲酸 | 5-Sulfoisophthalic acid
- CAS号:22326-31-4
- 别名:5-Sulfobenzene-1,3-dicarboxylic acid
- 分子式:C8H6O7S
- 分子量:246.19
- EINESC号:244-912-9
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Carnitine conjugate of nipecotic acid: a new example of dual prodrug.Carmela Napolitano et al.Molecules (Basel, Switzerland), 14(9), 3268-3274 (2009-09-29)
Anticonvulsant and anxiolytic activity of FrPbAII, a novel GABA uptake inhibitor isolated from the venom of the social spider Parawixia bistriata (Araneidae: Araneae).José Luiz Liberato et al.Brain research, 1124(1), 19-27 (2006-11-11)
Developmental control of spike-timing-dependent plasticity by tonic GABAergic signaling in striatum.Silvana Valtcheva et al.Neuropharmacology, 121, 261-277 (2017-04-15)
Synaptosomal GABA uptake decreases in paraoxon-treated rat brain.Moslem Mohammadi et al.Toxicology, 244(1), 42-48 (2007-12-07)
Determination of enantiomeric excess of nipecotic acid as 1-(7-nitrobenzo[c][1,2,5]oxadiazol-4-yl) derivatives.Simone K Schmidt et al.Chirality, 29(1), 48-56 (2016-12-27)
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Developmental Changes in Serotonergic Modulation of GABAergic Synaptic Transmission and Postsynaptic GABAA Receptor Composition in the Cerebellar Nuclei.Fumihito Saitow et al.Cerebellum (London, England), 17(3), 346-358 (2018-01-20)
VPACDiana Cunha-Reis et al.British journal of pharmacology, 174(24), 4725-4737 (2017-09-26)
N-methyl phenylalanine-rich peptides as highly versatile blood-brain barrier shuttles.Morteza Malakoutikhah et al.Journal of medicinal chemistry, 53(6), 2354-2363 (2010-02-23)
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Azetidine derivatives as novel gamma-aminobutyric acid uptake inhibitors: synthesis, biological evaluation, and structure-activity relationship.Mark R Faust et al.European journal of medicinal chemistry, 45(6), 2453-2466 (2010-03-12)
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Histamine H3 receptor activation counteracts adenosine A2A receptor-mediated enhancement of depolarization-evoked [3H]-GABA release from rat globus pallidus synaptosomes.Guadalupe-Elide Morales-Figueroa et al.ACS chemical neuroscience, 5(8), 637-645 (2014-06-03)
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: design, synthesis, and structure-activity relationships.Shigeo Hayashi et al.Bioorganic & medicinal chemistry, 18(21), 7675-7699 (2010-09-30)
GABA uptake transporters support dopamine release in dorsal striatum with maladaptive downregulation in a parkinsonism model.Bradley M Roberts et al.Nature communications, 11(1), 4958-4958 (2020-10-04)
Pharmacological identification of a guanidine-containing β-alanine analogue with low micromolar potency and selectivity for the betaine/GABA transporter 1 (BGT1).Anas Al-Khawaja et al.Neurochemical research, 39(10), 1988-1996 (2014-05-24)
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Synthesis and evaluation of N-substituted nipecotic acid derivatives with an unsymmetrical bis-aromatic residue attached to a vinyl ether spacer as potential GABA uptake inhibitors.Gabriele Quandt et al.Bioorganic & medicinal chemistry, 21(11), 3363-3378 (2013-04-20)
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Selective amino acid substitutions convert the creatine transporter to a gamma-aminobutyric acid transporter.Joanna R Dodd et al.The Journal of biological chemistry, 282(21), 15528-15533 (2007-04-03)
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Adenosine A2A Receptor Modulates the Activity of Globus Pallidus Neurons in Rats.Hui-Ling Diao et al.Frontiers in physiology, 8, 897-897 (2017-11-23)
GABAergic and glycinergic inhibitory mechanisms in the lamprey respiratory control.Fulvia Bongianni et al.Brain research, 1090(1), 134-145 (2006-04-25)
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Enduring changes in tonic GABAA receptor signaling in dentate granule cells after controlled cortical impact brain injury in mice.Jeffery A Boychuk et al.Experimental neurology, 277, 178-189 (2016-01-17)
Simultaneous determination of vigabatrin and amino acid neurotransmitters in brain microdialysates by capillary electrophoresis with laser-induced fluorescence detection.Nadia Benturquia et al.Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 806(2), 237-244 (2004-06-03)
Synthesis and biological evaluation of (R)-N-(diarylmethylthio/sulfinyl)ethyl/propyl-piperidine-3-carboxylic acid hydrochlorides as novel GABA uptake inhibitors.Jiange Zhang et al.Bioorganic & medicinal chemistry letters, 17(13), 3769-3773 (2007-05-23)
Chemical genetics reveals a complex functional ground state of neural stem cells.Phedias Diamandis et al.Nature chemical biology, 3(5), 268-273 (2007-04-10)
Inhibition of the uptake of GABA and related amino acids in rat brain slices by the optical isomers of nipecotic acid.G A Johnston et al.Journal of neurochemistry, 26(5), 1029-1032 (1976-05-01)
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