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Male contraception: history and development.Paul Kogan et al.The Urologic clinics of North America, 41(1), 145-161 (2013-11-30) Recent studies on lonidamine, the lead compound of the antispermatogenic indazol-carboxylic acids.Maria Teresa Gatto et al.Contraception, 65(4), 277-278 (2002-05-22) The fourth isoform of the adenine nucleotide translocator inhibits mitochondrial apoptosis in cancer cells.Cindy Gallerne et al.The international journal of biochemistry & cell biology, 42(5), 623-629 (2010-01-12) Glycosyl and polyalcoholic prodrugs of lonidamine.G Giorgioni et al.Bioorganic & medicinal chemistry letters, 18(7), 2445-2450 (2008-03-07) Combined modality clinical trials for favorable B-cell neoplasms: lonidamine plus whole body hyperthermia and/or total body irradiation.H I Robins Seminars in oncology, 18(2 Suppl 4), 23-27 (1991-04-01) Emerging drug therapies for benign prostatic hyperplasia.Travis L Bullock et al.Expert opinion on emerging drugs, 11(1), 111-123 (2006-03-01) The 18-kDa translocator protein (TSPO) disrupts mammary epithelial morphogenesis and promotes breast cancer cell migration.Xiaoting Wu et al.PloS one, 8(8), e71258-e71258 (2013-08-24) A novel effect of DMOG on cell metabolism: direct inhibition of mitochondrial function precedes HIF target gene expression.Alexander V Zhdanov et al.Biochimica et biophysica acta, 1847(10), 1254-1266 (2015-07-06) Utilizing Synergistic Potential of Mitochondria-Targeting Drugs for Leukemia Therapy.Svetlana B Panina et al.Frontiers in oncology, 10, 435-435 (2020-04-23) Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity.Marilisa P Dimmito et al.Biomolecules, 9(9) (2019-09-19) KMT2D Deficiency Impairs Super-Enhancers to Confer a Glycolytic Vulnerability in Lung Cancer.Hunain Alam et al.Cancer cell, 37(4), 599-617 (2020-04-04) Monoamine carboxylate transporters are involved in BI-1-associated cancer metastasis in HT1080 colon fibrosarcoma cells.Geum-Hwa Lee et al.International journal of oncology, 39(1), 209-216 (2011-05-04) Lonidamine: in vitro/in vivo correlations.B A Teicher European journal of cancer (Oxford, England : 1990), 30A(10), 1411-1413 (1994-01-01) Lonidamine in malignant brain tumors.D Schiffer et al.Seminars in oncology, 18(2 Suppl 4), 38-41 (1991-04-01) Curcumin stimulates reactive oxygen species production and potentiates apoptosis induction by the antitumor drugs arsenic trioxide and lonidamine in human myeloid leukemia cell lines.Yolanda Sánchez et al.The Journal of pharmacology and experimental therapeutics, 335(1), 114-123 (2010-07-08) Lonidamine in head and neck cancer: an overview.C W Scarantino et al.Seminars in oncology, 18(2 Suppl 4), 28-32 (1991-04-01) Targeting Cellular Metabolism in Acute Myeloid Leukemia and The Role of Patient Heterogeneity.Ida Sofie Grønningsæter et al.Cells, 9(5) (2020-05-13) Chemosensitization by knockdown of adenine nucleotide translocase-2.Morgane Le Bras et al.Cancer research, 66(18), 9143-9152 (2006-09-20) Development of a yeast bio-assay to screen anti-mitochondrial drugs.Johan L F Kock et al.Current drug discovery technologies, 6(3), 186-191 (2009-06-06) Increased apoptotic efficacy of lonidamine plus arsenic trioxide combination in human leukemia cells. Reactive oxygen species generation and defensive protein kinase (MEK/ERK, Akt/mTOR) modulation.Eva Calviño et al.Biochemical pharmacology, 82(11), 1619-1629 (2011-09-06) Lonidamine and related compounds.B Silvestrini et al.Progress in medicinal chemistry, 21, 110-135 (1984-01-01) Optimizing radiotherapy of brain tumours by a combination of temozolomide & lonidamine.S Prabhakara et al.The Indian journal of medical research, 128(2), 140-148 (2008-11-13) (31) P and (1) H MRS of DB-1 melanoma xenografts: lonidamine selectively decreases tumor intracellular pH and energy status and sensitizes tumors to melphalan.Kavindra Nath et al.NMR in biomedicine, 26(1), 98-105 (2012-06-30) A bioenergetic shift is required for spermatogonial differentiation.Wei Chen et al.Cell discovery, 6, 56-56 (2020-08-31) Does granulocyte colony-stimulating factor worsen anemia in early breast cancer patients treated with epirubicin and cyclophosphamide?Paola Papaldo et al.Journal of clinical oncology : official journal of the American Society of Clinical Oncology, 24(19), 3048-3055 (2006-06-14) Lonidamine affects testicular steroid hormones in immature mice.Maria Elsa Traina et al.Toxicology and applied pharmacology, 221(1), 95-101 (2007-04-20) Development of EGFR-targeted polymer blend nanocarriers for combination paclitaxel/lonidamine delivery to treat multi-drug resistance in human breast and ovarian tumor cells.Lara Milane et al.Molecular pharmaceutics, 8(1), 185-203 (2010-10-15) Development of targeting lonidamine liposomes that circumvent drug-resistant cancer by acting on mitochondrial signaling pathways.Nan Li et al.Biomaterials, 34(13), 3366-3380 (2013-02-16) Toxicity and clinical tolerance of lonidamine.G Robustelli della Cuna et al.Seminars in oncology, 18(2 Suppl 4), 18-22 (1991-04-01) [Treatment and post-treatment with lonidamine in human colon carcinoma HT-29 cell line].Alicia G Fuchs Medicina, 68(1), 13-22 (2008-04-18) Curcumin stimulates reactive oxygen species production and potentiates apoptosis induction by the antitumor drugs arsenic trioxide and lonidamine in human myeloid leukemia cell lines.Yolanda Sánchez et al.The Journal of pharmacology and experimental therapeutics, 335(1), 114-123 (2010-07-08) Lonidamine in head and neck cancer: an overview.C W Scarantino et al.Seminars in oncology, 18(2 Suppl 4), 28-32 (1991-04-01) Recent studies on lonidamine, the lead compound of the antispermatogenic indazol-carboxylic acids.Maria Teresa Gatto et al.Contraception, 65(4), 277-278 (2002-05-22) The fourth isoform of the adenine nucleotide translocator inhibits mitochondrial apoptosis in cancer cells.Cindy Gallerne et al.The international journal of biochemistry & cell biology, 42(5), 623-629 (2010-01-12) Glycosyl and polyalcoholic prodrugs of lonidamine.G Giorgioni et al.Bioorganic & medicinal chemistry letters, 18(7), 2445-2450 (2008-03-07) Combined modality clinical trials for favorable B-cell neoplasms: lonidamine plus whole body hyperthermia and/or total body irradiation.H I Robins Seminars in oncology, 18(2 Suppl 4), 23-27 (1991-04-01) Emerging drug therapies for benign prostatic hyperplasia.Travis L Bullock et al.Expert opinion on emerging drugs, 11(1), 111-123 (2006-03-01) The 18-kDa translocator protein (TSPO) disrupts mammary epithelial morphogenesis and promotes breast cancer cell migration.Xiaoting Wu et al.PloS one, 8(8), e71258-e71258 (2013-08-24) A novel effect of DMOG on cell metabolism: direct inhibition of mitochondrial function precedes HIF target gene expression.Alexander V Zhdanov et al.Biochimica et biophysica acta, 1847(10), 1254-1266 (2015-07-06) Utilizing Synergistic Potential of Mitochondria-Targeting Drugs for Leukemia Therapy.Svetlana B Panina et al.Frontiers in oncology, 10, 435-435 (2020-04-23) Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity.Marilisa P Dimmito et al.Biomolecules, 9(9) (2019-09-19) KMT2D Deficiency Impairs Super-Enhancers to Confer a Glycolytic Vulnerability in Lung Cancer.Hunain Alam et al.Cancer cell, 37(4), 599-617 (2020-04-04) Monoamine carboxylate transporters are involved in BI-1-associated cancer metastasis in HT1080 colon fibrosarcoma cells.Geum-Hwa Lee et al.International journal of oncology, 39(1), 209-216 (2011-05-04) Lonidamine: in vitro/in vivo correlations.B A Teicher European journal of cancer (Oxford, England : 1990), 30A(10), 1411-1413 (1994-01-01) Lonidamine in malignant brain tumors.D Schiffer et al.Seminars in oncology, 18(2 Suppl 4), 38-41 (1991-04-01) Aerobic glycolysis tunes YAP/TAZ transcriptional activity.Elena Enzo et al.The EMBO journal, 34(10), 1349-1370 (2015-03-23) Male contraception: history and development.Paul Kogan et al.The Urologic clinics of North America, 41(1), 145-161 (2013-11-30) Targeting Cellular Metabolism in Acute Myeloid Leukemia and The Role of Patient Heterogeneity.Ida Sofie Grønningsæter et al.Cells, 9(5) (2020-05-13) Chemosensitization by knockdown of adenine nucleotide translocase-2.Morgane Le Bras et al.Cancer research, 66(18), 9143-9152 (2006-09-20) Development of a yeast bio-assay to screen anti-mitochondrial drugs.Johan L F Kock et al.Current drug discovery technologies, 6(3), 186-191 (2009-06-06) Increased apoptotic efficacy of lonidamine plus arsenic trioxide combination in human leukemia cells. Reactive oxygen species generation and defensive protein kinase (MEK/ERK, Akt/mTOR) modulation.Eva Calviño et al.Biochemical pharmacology, 82(11), 1619-1629 (2011-09-06) Lonidamine and related compounds.B Silvestrini et al.Progress in medicinal chemistry, 21, 110-135 (1984-01-01) Optimizing radiotherapy of brain tumours by a combination of temozolomide & lonidamine.S Prabhakara et al.The Indian journal of medical research, 128(2), 140-148 (2008-11-13) (31) P and (1) H MRS of DB-1 melanoma xenografts: lonidamine selectively decreases tumor intracellular pH and energy status and sensitizes tumors to melphalan.Kavindra Nath et al.NMR in biomedicine, 26(1), 98-105 (2012-06-30) A bioenergetic shift is required for spermatogonial differentiation.Wei Chen et al.Cell discovery, 6, 56-56 (2020-08-31) Does granulocyte colony-stimulating factor worsen anemia in early breast cancer patients treated with epirubicin and cyclophosphamide?Paola Papaldo et al.Journal of clinical oncology : official journal of the American Society of Clinical Oncology, 24(19), 3048-3055 (2006-06-14) Lonidamine affects testicular steroid hormones in immature mice.Maria Elsa Traina et al.Toxicology and applied pharmacology, 221(1), 95-101 (2007-04-20) Development of EGFR-targeted polymer blend nanocarriers for combination paclitaxel/lonidamine delivery to treat multi-drug resistance in human breast and ovarian tumor cells.Lara Milane et al.Molecular pharmaceutics, 8(1), 185-203 (2010-10-15) Development of targeting lonidamine liposomes that circumvent drug-resistant cancer by acting on mitochondrial signaling pathways.Nan Li et al.Biomaterials, 34(13), 3366-3380 (2013-02-16) Toxicity and clinical tolerance of lonidamine.G Robustelli della Cuna et al.Seminars in oncology, 18(2 Suppl 4), 18-22 (1991-04-01)

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