密度	1.284

没有数据	没有数据

来源	SDS样本
没有数据	没有数据

产品合成路线

更多

名称	CAS号

更多

文章

同行评议文献

[Cardiac, respiratory, and motor activity in norm and after activation of catecholaminergic systems in newborn rat pups].S V Kuznetsov et al.Zhurnal evoliutsionnoi biokhimii i fiziologii, 48(4), 367-379 (2012-09-28) The pharmacology of sulpiride--a dopamine receptor antagonist.S E O'Connor et al.General pharmacology, 13(3), 185-193 (1982-01-01) Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.G Okugawa et al.Journal of neuroendocrinology, 11(11), 887-895 (1999-10-16) Successful treatment of atypical depression with amisulpride: a case report.Sri M Agarwal et al.Asian journal of psychiatry, 5(4), 362-362 (2012-11-24) [The benzamides tiapride, sulpiride, and amisulpride in treatment for Tourette's syndrome].K R Müller-Vahl Der Nervenarzt, 78(3), 264-264 (2006-08-23) Exploring the role of different drug transport routes in permeability screening.Pär Matsson et al.Journal of medicinal chemistry, 48(2), 604-613 (2005-01-22) A 6-week, randomized, multicentre, open-label study comparing efficacy and tolerability of amisulpride at a starting dose of 400 mg/day versus 800 mg/day in patients with acute exacerbations of schizophrenia.Seung Jae Lee et al.Clinical drug investigation, 32(11), 735-745 (2012-09-29) [Toxicity of sulpiride].Krzysztof Ciszowski et al.Przeglad lekarski, 67(8), 606-609 (2010-01-01) Sulpiride: an antipsychotic with selective dopaminergic antagonist properties.C F Caley et al.The Annals of pharmacotherapy, 29(2), 152-160 (1995-02-01) A risk-benefit assessment of sulpiride in the treatment of schizophrenia.M C Mauri et al.Drug safety, 14(5), 288-298 (1996-05-01) Orexin A induced antinociception in the ventral tegmental area involves D1 and D2 receptors in the nucleus accumbens.Saeid Yazdi-Ravandi et al.Pharmacology, biochemistry, and behavior, 126, 1-6 (2014-09-03) Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates.Semra Isik et al.Bioorganic & medicinal chemistry, 17(3), 1158-1163 (2009-01-07) [Possibilities in using sulpiride in the treatment of psychotic disorders].D S Danilov Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova, 112(6), 91-97 (2012-09-18) Blocking Dopaminergic Signaling Soon after Learning Impairs Memory Consolidation in Guinea Pigs.Kiera-Nicole Lee et al.PloS one, 10(8), e0135578-e0135578 (2015-08-15) Spectroscopic investigation on the inclusion complex formation between amisulpride and γ-cyclodextrin.Jeetendra Singh Negi et al.Carbohydrate polymers, 92(2), 1835-1843 (2013-02-13) Dopamine D1 or D2 receptor blockade in the globus pallidus produces akinesia in the rat.W Hauber et al.Behavioural brain research, 106(1-2), 143-150 (1999-12-14) [A case of male infertility caused by drug-induced hyperprolactinemia].Teppei Takeshima et al.Hinyokika kiyo. Acta urologica Japonica, 59(1), 65-67 (2013-02-16) Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.Denis Fourches et al.Chemical research in toxicology, 23(1), 171-183 (2009-12-18) I.V. APD421 (amisulpride) prevents postoperative nausea and vomiting: a randomized, double-blind, placebo-controlled, multicentre trial.P Kranke et al.British journal of anaesthesia, 111(6), 938-945 (2013-07-23) The relation between symptom improvement and gastric emptying in the treatment of diabetic and idiopathic gastroparesis.Pieter Janssen et al.The American journal of gastroenterology, 108(9), 1382-1391 (2013-09-06) Delusional infestation: a clinical profile.M S Bhatia et al.Asian journal of psychiatry, 6(2), 124-127 (2013-03-08) Antagonism by haloperidol and its metabolites of mechanical hypersensitivity induced by intraplantar capsaicin in mice: role of sigma-1 receptors.José M Entrena et al.Psychopharmacology, 205(1), 21-33 (2009-03-28) Dopamine D2 receptor stimulation differentially affects voltage-activated calcium channels in rat pituitary melanotropic cells.J A Keja et al.The Journal of physiology, 450, 409-435 (1992-05-01) Neurotensin Induces Presynaptic Depression of D2 Dopamine Autoreceptor-Mediated Neurotransmission in Midbrain Dopaminergic Neurons.Elisabeth Piccart et al.The Journal of neuroscience : the official journal of the Society for Neuroscience, 35(31), 11144-11152 (2015-08-08) Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs?Daniela Vullo et al.Bioorganic & medicinal chemistry letters, 15(4), 963-969 (2005-02-03) Improvements in micturition and urinary retention after switching from amisulpiride to paliperidone in a schizophrenic patient.Chien-Han Lai The Journal of neuropsychiatry and clinical neurosciences, 24(4), E11-E12 (2012-12-12) Anaphylaxis due to sulpiride and sensitization to metamizole.M I Alvarado et al.Journal of investigational allergology & clinical immunology, 22(5), 379-380 (2012-10-30) Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors.Isao Nishimori et al.Journal of medicinal chemistry, 48(24), 7860-7866 (2005-11-24) The effect of cholestasis on rewarding and exploratory behaviors induced by opioidergic and dopaminergic agents in mice.Mohaddeseh Ebrahimi-ghiri et al.Archives of Iranian medicine, 15(10), 617-624 (2012-10-02) Carbonic anhydrase inhibitors: Hypoxia-activatable sulfonamides incorporating disulfide bonds that target the tumor-associated isoform IX.Giuseppina De Simone et al.Journal of medicinal chemistry, 49(18), 5544-5551 (2006-09-01) Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana.Anna Ohradanova et al.Bioorganic & medicinal chemistry, 20(4), 1403-1410 (2012-01-31) Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.G Okugawa et al.Journal of neuroendocrinology, 11(11), 887-895 (1999-10-16) Neural computational prediction of oral drug absorption based on CODES 2D descriptors.A Guerra et al.European journal of medicinal chemistry, 45(3), 930-940 (2009-12-22) Antipsychotic combination using low-dose antipsychotics is as efficacious and safe as, but cheaper, than optimal-dose monotherapy in the treatment of schizophrenia: a randomized, double-blind study.Ching-Hua Lin et al.International clinical psychopharmacology, 28(5), 267-274 (2013-06-20) [A case of male infertility caused by drug-induced hyperprolactinemia].Teppei Takeshima et al.Hinyokika kiyo. Acta urologica Japonica, 59(1), 65-67 (2013-02-16) Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.Denis Fourches et al.Chemical research in toxicology, 23(1), 171-183 (2009-12-18) Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates.Semra Isik et al.Bioorganic & medicinal chemistry, 17(3), 1158-1163 (2009-01-07) [Changes in the endocrine system in the course of sulpiride therapy].L T Roś Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego, 11(66), 532-534 (2002-03-20) Changes on D2-like receptor induced Gi protein activation and hippocampal dopamine release in kindled rats.David Alcantara-Gonzalez et al.Progress in neuro-psychopharmacology & biological psychiatry, 40, 246-251 (2012-10-23) Cloning, characterization, and inhibition studies of a beta-carbonic anhydrase from Brucella suis.Pascale Joseph et al.Journal of medicinal chemistry, 53(5), 2277-2285 (2010-02-18) Social feeding in Caenorhabditis elegans is modulated by antipsychotic drugs and calmodulin and may serve as a protophenotype for asociality.Donard S Dwyer et al.Neuropharmacology, 92, 56-62 (2015-01-13) [Metoclopramide, sulpiride, and chlorpromazine loading test].K Azuma et al.Nihon rinsho. Japanese journal of clinical medicine, 55 Suppl 2, 249-251 (1997-04-01) Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties.M Amelia Santos et al.Bioorganic & medicinal chemistry letters, 17(6), 1538-1543 (2007-01-26) Identifying clinically meaningful symptom response cut-off values on the SANS in predominant negative symptoms.Stephen Z Levine et al.Schizophrenia research, 145(1-3), 125-127 (2013-02-12) I.V. APD421 (amisulpride) prevents postoperative nausea and vomiting: a randomized, double-blind, placebo-controlled, multicentre trial.P Kranke et al.British journal of anaesthesia, 111(6), 938-945 (2013-07-23) Physicochemical determinants of human renal clearance.Manthena V S Varma et al.Journal of medicinal chemistry, 52(15), 4844-4852 (2009-05-19) Development of an in silico model for human skin permeation based on a Franz cell skin permeability assay.Pil H Lee et al.Bioorganic & medicinal chemistry letters, 20(1), 69-73 (2009-12-08) Dopamine modulates persistent synaptic activity and enhances the signal-to-noise ratio in the prefrontal cortex.Sven Kroener et al.PloS one, 4(8), e6507-e6507 (2009-08-06) Chemical genetics reveals a complex functional ground state of neural stem cells.Phedias Diamandis et al.Nature chemical biology, 3(5), 268-273 (2007-04-10) Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors.Isao Nishimori et al.Journal of medicinal chemistry, 50(2), 381-388 (2007-01-19) Cortically driven Fos induction in the striatum is amplified by local dopamine D2-class receptor blockade.S Berretta et al.The European journal of neuroscience, 11(12), 4309-4319 (1999-12-14) Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.Fabrizio Carta et al.Bioorganic & medicinal chemistry letters, 19(23), 6649-6654 (2009-10-23) Involvement of dopaminergic receptors of the rat nucleus accumbens in decreasing the conditioned place preference induced by lateral hypothalamus stimulation.Abbas Haghparast et al.Neuroscience letters, 556, 10-14 (2013-10-10) Dopamine receptor activation increases HIV entry into primary human macrophages.Peter J Gaskill et al.PloS one, 9(9), e108232-e108232 (2014-10-01) Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata.Anthony Bertucci et al.Bioorganic & medicinal chemistry letters, 21(2), 710-714 (2011-01-07) A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth.Pascale Joseph et al.Bioorganic & medicinal chemistry, 19(3), 1172-1178 (2011-01-22) Carbonic anhydrase inhibitors. Inhibition and homology modeling studies of the fungal beta-carbonic anhydrase from Candida albicans with sulfonamides.Alessio Innocenti et al.Bioorganic & medicinal chemistry, 17(13), 4503-4509 (2009-05-20) Abnormal modulation of reward versus punishment learning by a dopamine D2-receptor antagonist in pathological gamblers.Lieneke Katharina Janssen et al.Psychopharmacology, 232(18), 3345-3353 (2015-06-21) Charles Bonnet syndrome responding to amisulpride.M S Bhatia et al.The Journal of neuropsychiatry and clinical neurosciences, 24(3), E40-E40 (2012-10-06) Cloning, expression, post-translational modifications and inhibition studies on the latest mammalian carbonic anhydrase isoform, CA XV.Mika Hilvo et al.Journal of medicinal chemistry, 52(3), 646-654 (2009-02-06) Cognitive effects of a single dose of atypical antipsychotics in healthy volunteers compared with placebo or haloperidol.Young-Chul Chung et al.Journal of clinical psychopharmacology, 32(6), 778-786 (2012-11-08) [Sulpiride: an atypical neuroleptic with a wide spectrum of therapeutic claims].A Wasieczko et al.Psychiatria polska, 30(6), 1009-1016 (1996-11-01) Citalopram and levosulpiride: a dangerous drug combination for QT prolongation.Sergio Agosti et al.The American journal of emergency medicine, 31(11), 1624-1624 (2013-07-31) Toxicological screening of human plasma by on-line SPE-HPLC-DAD: identification and quantification of basic drugs and metabolites.Ludmila Mut et al.Biomedical chromatography : BMC, 29(6), 935-952 (2014-11-18) Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.Isao Nishimori et al.Journal of medicinal chemistry, 49(6), 2117-2126 (2006-03-17) Light-dependent translocation of arrestin in rod photoreceptors is signaled through a phospholipase C cascade and requires ATP.Wilda Orisme et al.Cellular signalling, 22(3), 447-456 (2009-11-06) Punishment-induced behavioral and neurophysiological variability reveals dopamine-dependent selection of kinematic movement parameters.Joseph M Galea et al.The Journal of neuroscience : the official journal of the Society for Neuroscience, 33(9), 3981-3988 (2013-03-01) Antidepressant-like activity of ellagic acid in unstressed and acute immobilization-induced stressed mice.Dinesh Dhingra et al.Pharmacological reports : PR, 64(4), 796-807 (2012-10-23) Expanding Role of Dopaminergic Inhibition in Hypercapnic Responses of Cultured Rat Carotid Body Cells: Involvement of Type II Glial Cells.Erin M Leonard et al.International journal of molecular sciences, 21(15) (2020-08-06) In silico Analysis of Sulpiride, Synthesis, Characterization and In vitro Studies of its Nanoparticle for the Treatment of Schizophrenia.Serda Kecel-Gunduz et al.Current computer-aided drug design, 16(2), 104-121 (2019-06-28) Hypolipidemic and weight reducing activity of the ethanolic extract of Tamarindus indica fruit pulp in cafeteria diet- and sulpiride-induced obese rats.Vaneeta Jindal et al.Journal of pharmacology & pharmacotherapeutics, 2(2), 80-84 (2011-07-21) Hypothalamic Prolactin Regulation of Luteinizing Hormone Secretion in the Female Rat.Pasha Grachev et al.Endocrinology, 156(8), 2880-2892 (2015-05-21) Carbonic anhydrase inhibitors: the beta-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitors.Isao Nishimori et al.Bioorganic & medicinal chemistry letters, 17(13), 3585-3594 (2007-05-08) Optimizing Multiple Analyte Injections in Surface Plasmon Resonance Biosensors with Analytes having Different Refractive Index Increments.Massinissa Si Mehand et al.Scientific reports, 5, 15855-15855 (2015-10-31) Mismatch negativity and cognitive performance for the prediction of psychosis in subjects with at-risk mental state.Yuko Higuchi et al.PloS one, 8(1), e54080-e54080 (2013-01-26) Validated spectrofluorimetric method for determination of sulpiride in commercial formulations using Hantzsch condensation reaction.Jasmin Shah et al.Pakistan journal of pharmaceutical sciences, 26(5), 921-928 (2013-09-17) Sulpiride augmentation for schizophrenia.Jijun Wang et al.Schizophrenia bulletin, 36(2), 229-230 (2010-01-12) Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.Manthena V S Varma et al.Journal of medicinal chemistry, 53(3), 1098-1108 (2010-01-15) Sulpiride augmentation in people with schizophrenia partially responsive to clozapine. A double-blind, placebo-controlled study.R Shiloh et al.The British journal of psychiatry : the journal of mental science, 171, 569-573 (1998-03-31) The mode of action of sulpiride as an atypical antidepressant agent.P Jenner et al.Advances in biochemical psychopharmacology, 32, 85-103 (1982-01-01) Possible mechanism of antidepressant effect of L-sulpiride.G Serra et al.Clinical neuropharmacology, 13 Suppl 1, S76-S83 (1990-01-01) Loss of feedback inhibition via D2 autoreceptors enhances acquisition of cocaine taking and reactivity to drug-paired cues.Kathryn B Holroyd et al.Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 40(6), 1495-1509 (2014-12-31) In-situ forming gel-like depot of a polyaspartamide-polylactide copolymer for once a week administration of sulpiride.Calogero Fiorica et al.The Journal of pharmacy and pharmacology, 67(1), 78-86 (2014-09-23) Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori.Isao Nishimori et al.Bioorganic & medicinal chemistry letters, 16(8), 2182-2188 (2006-02-07) Poisoning: fact or fiction?Robert J Flanagan The Medico-legal journal, 80(Pt 4), 127-148 (2013-01-24) Augmentation with sulpiride for a schizophrenic patient partially responsive to clozapine.J H Stubbs et al.Acta psychiatrica Scandinavica, 102(5), 390-393 (2000-12-01) Preparation and pharmacological characterization of trans-2-amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes as D2-like dopamine receptor agonists.Antonio Di Stefano et al.Journal of medicinal chemistry, 48(7), 2646-2654 (2005-04-02) Intrahippocampal administration of D2 but not D1 dopamine receptor antagonist suppresses the expression of conditioned place preference induced by morphine in the ventral tegmental area.Abbas Haghparast et al.Neuroscience letters, 541, 138-143 (2013-03-19) [Sulpiride: the best known atypical, safe neuroleptic drug. Review of literature].M Rzewuska Psychiatria polska, 32(5), 655-666 (1999-01-28) [Antiemetic properties of levo-sulpiride].M Guslandi Minerva medica, 81(12), 855-860 (1990-12-01) Diagnostic exercise.V M Lucke et al.Laboratory animal science, 29(5), 601-602 (1979-10-01) Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.Xiaofan Sui et al.European journal of medicinal chemistry, 44(11), 4455-4460 (2009-07-10) Sulpiride versus placebo for schizophrenia.Ichiro M Omori et al.The Cochrane database of systematic reviews, (2)(2), CD007811-CD007811 (2009-04-17) [The comparative study on the efficacy of the combination of serotonin reuptake inhibitor antidepressants and antipsychotics in the treatment of recurrent depressive disorders].A L D'iakonov et al.Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova, 112(11 Pt 2), 61-66 (2012-12-22) Effects of dopaminergic agents on progression of naturally occurring myopia in albino guinea pigs (Cavia porcellus).Liqin Jiang et al.Investigative ophthalmology & visual science, 55(11), 7508-7519 (2014-10-02) Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates.Isao Nishimori et al.Bioorganic & medicinal chemistry, 19(16), 5023-5030 (2011-07-16) Attaining and sustaining remission of predominant negative symptoms.Stephen Z Levine et al.Schizophrenia research, 143(1), 60-64 (2012-12-12) Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides.Anthony Bertucci et al.Bioorganic & medicinal chemistry, 17(14), 5054-5058 (2009-06-13) QSAR-based permeability model for drug-like compounds.Rafael Gozalbes et al.Bioorganic & medicinal chemistry, 19(8), 2615-2624 (2011-04-05) Safety of the electroconvulsive therapy and amisulpride combination.Rozália Takács et al.Psychiatria Danubina, 25(1), 76-79 (2013-03-09) Sulpiride for schizophrenia.B G Soares et al.The Cochrane database of systematic reviews, (2)(2), CD001162-CD001162 (2000-05-05) Protein kinase C beta regulates the D₂-like dopamine autoreceptor.Kathryn D Luderman et al.Neuropharmacology, 89, 335-341 (2014-12-03) Sulpiride augmentation for schizophrenia.Jijun Wang et al.The Cochrane database of systematic reviews, (1)(1), CD008125-CD008125 (2010-01-22) Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis.Isao Nishimori et al.Journal of medicinal chemistry, 52(9), 3116-3120 (2009-04-03) Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).Giulia Caron et al.Journal of medicinal chemistry, 48(9), 3269-3279 (2005-04-29) [Schizophrenia-like psychotic symptoms in a patient with confirmed Huntington's disease: a case report].Bartosz Grabski et al.Psychiatria polska, 46(4), 665-675 (2012-12-12) Improvement of ketamine-induced social withdrawal in rats: the role of 5-HT7 receptors.Małgorzata Hołuj et al.Behavioural pharmacology, 26(8 Spec No), 766-775 (2015-03-15) Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.Yun W Alelyunas et al.Bioorganic & medicinal chemistry letters, 20(24), 7312-7316 (2010-11-09) Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.Lei Du-Cuny et al.Bioorganic & medicinal chemistry, 17(19), 6983-6992 (2009-09-08) [Effect of antipsychotic amisulpride on immune reactivity].G V Idova et al.Eksperimental'naia i klinicheskaia farmakologiia, 76(5), 14-17 (2013-08-02) Ethanol-mediated facilitation of AMPA receptor function in the dorsomedial striatum: implications for alcohol drinking behavior.Jun Wang et al.The Journal of neuroscience : the official journal of the Society for Neuroscience, 32(43), 15124-15132 (2012-10-27) Prediction of drug intestinal absorption by new linear and non-linear QSPR.Alan Talevi et al.European journal of medicinal chemistry, 46(1), 218-228 (2010-11-30) Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes.Frank Boeckler et al.Journal of medicinal chemistry, 48(3), 694-709 (2005-02-04) Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.Johannes Kornhuber et al.Journal of medicinal chemistry, 51(2), 219-237 (2007-11-22) The Japanese toxicogenomics project: application of toxicogenomics.Takeki Uehara et al.Molecular nutrition & food research, 54(2), 218-227 (2009-12-31) Pharmacological assessment of methamphetamine-induced behavioral hyperactivity mediated by dopaminergic transmission in planarian Dugesia japonica.Natsuka Tashiro et al.Biochemical and biophysical research communications, 449(4), 412-418 (2014-05-27) Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides.Isao Nishimori et al.Bioorganic & medicinal chemistry, 15(23), 7229-7236 (2007-09-11)

备注